References

1.    Structure of the Prostaglandin H2 synthase-1 homo-dimer.   http://www.ks.uiuc.edu/

2.    Picot D, Loll PJ, Garavito RM.(1994) The X-ray crystal structure of the membrane protein prostaglandin H2 synthase-1. Nature  Jan 20;367(6460):243-9

3.   Smith WL, DeWitt DL. Biochemistry of prostaglandin endoperoxide H synthase-1 and synthase-2 and their differential susceptibility to nonsteroidal anti-inflammatory drugs. Semin Nephrol 1995 May;15(3):179-94

4.  The conversion of Arachidonic acid to Prostaglandins, prostacyclin and thromboxane A2. http://life.nthu.edu.tw/~g874214/final/text.html

5.  Picot D, Loll PJ, Garavito RM.  X-ray crystallographic study of the structure of prostaglandin H synthase. Adv Exp Med Biol 1997;400A:107-11

6.  PGHS-1 Peroxidase
http://gaea.bch.msu.edu/labs/garavito/web/index.htm

7.  Malkowski MG, Ginell SL, Smith WL, Garavito RM.  The productive conformation of arachidonic acid bound to prostaglandin synthase.Science 2000 Sep 15;289(5486):1933-7

8.  Loll PJ, Picot D, Ekabo O, Garavito RM. Synthesis and use of iodinated nonsteroidal antiinflammatory drug analogs as crystallographic probes of the prostaglandin H2 synthase cyclooxygenase active site.  Biochemistry 1996 Jun 11;35(23):7330-40

Rasmol references:

1.   Prostaglandin H2 synthase-1  Garavito RM, Picot D, Loll PJ. The 3.1 A X-ray crystal structure of the integral membrane enzyme prostaglandin H2 synthase-1. Adv Prostaglandin Thromboxane Leukot Res 1995;23:99-103

2.  Arachidonic acid (substrate) bound in the cyclooxygenase active site of PGHS-1  (chain A) (sheep)  Malkowski MG, Ginell SL, Smith WL, Garavito RM.  The productive conformation of arachidonic acid bound to prostaglandin synthase. Science 2000 Sep 15;289(5486):1933-7

3.  PGHS-1 complexed with the inhibitor P-(2'-iodo-5'-thenoyl)hydrotropic acid [Iodosuprofen].  Loll PJ, Picot D, Ekabo O, Garavito RM. Synthesis and use of iodinated nonsteroidal antiinflammatory drug analogs as crystallographic probes of the prostaglandin H2 synthase cyclooxygenase active site. Biochemistry 1996 Jun 11;35(23):7330-40 

 
 
 
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